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カタログ番号	製品名	別名	ターゲット
T0855	(R)-Naproxen		COX
	(R)-Naproxen, an anti-inflammatory agent, has antipyretic and analgesic properties. Both the acid and its sodium salt are used in the therapy of acute gout or dysmenorrhea, musculoskeletal disorders, rheumatoid arthritis...		COX
T21408	DM1-SMe	DM1-SSMe	Microtubule Associated
	DM1-SMe (DM1-SSMe) is a potent inhibitor of maytansinoid microtubular. DM1-SMe is about 3 to 10-fold more potent than the parent drug Maytansine, with IC50s of 0.003 to 0.01 nM for DM1-SMe in a panel of human tumor cell ...		Microtubule Associated
T12477	Uzansertib phosphate	INCB053914 phosphate	Pim
	Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase(PIM1, PIM2, PIM3 with IC50s of 0.24 nM, 30 nM, 0.12 nM , respectively).		Pim
TQ0059	Ilorasertib	ABT-348	VEGFR , FLT , c-RET , PDGFR , Aurora Kinase
	Ilorasertib (ABT-348) (ABT-348) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora A/Aurora B/Aurora C (IC50s: 120 nM/7 nM/1 nM). It also suppresses RET tyrosine kinase, PDGFRβ, and Flt1 (IC50s: ...		VEGFR , FLT , c-RET , PDGFR , Aurora Kinase
T6426	Buclizine dihydrochloride	Longifene,Buclina,Buclizine HCl,UCB-4445	5-HT Receptor , AChR , Histamine Receptor
	Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and antivertigo activities. Buclizine dihydrochloride binds to and ...		5-HT Receptor , AChR , Histamine Receptor
T6018	Zosuquidar trihydrochloride	Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride	P-gp
	Zosuquidar trihydrochloride (LY-335979 trihydrochloride) is a potent modulator of P-glycoprotein-mediated multi-drug resistance with Ki of 60 nM. Phase 3.		P-gp
T20864	7-Troc-paclitaxel		Others
	7-Troc-paclitaxel is a precursor of paclitaxel which has anti-tumor activity.		Others
T10342	Antitumor agent-2		Others
	Antitumor agent-2 has anti-inflammatory and anti-tumor activity and can be used to study cancer.		Others
T26623	AMRI-59	AMRI 59	Others
	AMRI-59 is a potent inhibitor of PrxI with anti-tumor activity.		Others
T12140	N-Acetyl-Calicheamicin	N-Acetyl-Calicheamicin γ,N-Acetyl-γ-calicheamicin	Antibacterial
	N-Acetyl-Calicheamicin (N-Acetyl-γ-calicheamicin) is an antibiotic with high anti-tumor activity.		Antibacterial
T23480	U-83836E		Others
	U-83836E (lazaroid ) has neuroprotective activity and anti-tumor activity, inhibits glioma cell proliferation, inhibits tumor necrosis factor and reverses endotoxin-induced shock.		Others
T3170	Troglitazone	CS-045,Romozin,Rezulin,Romglizone,Noscal,Prelay	Apoptosis , Ferroptosis , PPAR , Autophagy
	Troglitazone (Romglizone) is a PPARγ agonist with anti-inflammatory and anti-tumor activity.		Apoptosis , Ferroptosis , PPAR , Autophagy
T19783	Dehydroabiethylamine	NSC-2955,NSC 2955,Dehydroabietylamine,NSC2955,Leelamine free base,Leelamine	P450 , PDK
	Dehydroabiethylamine (NSC-2955) is an inducer of hepatic CYP2B activity. Dehydroabiethylamine inhibits pyruvate dehydrogenase kinases (PDKs) and intracellular cholesterol transport with anti-tumor activity.		P450 , PDK
T9027	CA-4948	Emavusertib	IRAK , FLT
	CA-4948 (Emavusertib) is a potent IRAK4/FLT3 inhibtor. CA-4948 with anti-tumor activity.		IRAK , FLT
T8340	Quinocetone		Others , Antibacterial , Antibiotic
	Quinocetone is an animal growth promoter and potential anti-tumor activity.		Others , Antibacterial , Antibiotic
TNU0085	2'-Deoxy-2'-fluoroarabinoadenosine		Nucleoside Antimetabolite/Analog
	2'-Deoxy-2'-fluoroarabinoadenosine is a nucleoside analogue with extensive anti-tumor activity and can be used for the study of tumor diseases.		Nucleoside Antimetabolite/Analog
T9582	CLEFMA		NF-κB
	CLEFMA has anti-proliferative activity. CLEFMA inhibits tumor growth associated with NF-κB-regulated anti-inflammatory and anti-metastatic effects.		NF-κB
T28424	PKUMDL-WQ-2101		Dehydrogenase
	PKUMDL-WQ-2101 is a selective allosteric inhibitor of phosphoglycerate dehydrogenase with anti-tumor activity.		Dehydrogenase
T20158	Phenformin	Debeone,N-Phenethylbiguanide,Insoral,BRN 1977317,Azucaps	Apoptosis
	Phenformin (BRN 1977317) is a biguanide compound with anticancer and anti-glycemic activity, inhibits skin tumor growth and promotes keratinocyte differentiation and apoptosis.		Apoptosis
T16936	SS-208		HDAC
	SS-208 is a selective inhibitor of HDAC6 (IC50 = 12 nM) with anti-tumor activity. SS-208 shows selectivity over other HDAC subtypes.		HDAC
T40286	KRAS G12C inhibitor 19		Ras
	KRAS G12C inhibitor 19 is a potent KRAS G12C inhibitor that shows anti-tumor activity in cellular assays, and the family inhibits tumor growth.		Ras
T78212	RMC-9805	KRAS G12D inhibitor 18,KRAS G12D IN 18	Others
	RMC-9805 is a potent KRAS G12D inhibitor with potential anti-tumor and inhibitory activity against tumor cell proliferation for the study of pancreatic cancer.		Others
T4360	ML385		Others , Ferroptosis , Nrf2
	ML385 is an NRF2 inhibitor (IC50=1.9 μM) with novelty and specificity. ML385 has anti-inflammatory activity by modulating anti-oxidative stress through the inhibition of NRF2. ML385 also exhibits anti-tumor activity.		Others , Ferroptosis , Nrf2
T8843	APS6-45		MAPK , Ras
	APS6-45 inhibits RAS/MAPK signaling and exhibits anti-tumor activity.		MAPK , Ras
T65550	Gefitinib analog III	4-((3-Chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl acetate	Others
	Gefitinib analog III (4-((3-Chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl acetate) has potential anti-inflammatory and anti-tumor activity and can be used to study its interactions and activity in organisms.		Others
T11666	IPR-803		Serine/threonin kinase
	IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity. IPR-803 binds directly to uPAR with a Ki of 0.2 μM.		Serine/threonin kinase
T15793	Lurbinectedin	PM01183	Others
	Lurbinectedin (PM01183) is a DNA minor groove covalent binder. Lurbinectedin also shows effective anti-tumor activity.		Others
T12246	CB-103		Gamma-secretase
	CB-103 is a orally active inhibitor of notch signaling pathway, with anti-tumor activity.		Gamma-secretase
T63518	USP1-IN-2		DUB
	USP1-IN-2 is a potent USP1 inhibitor with potential anti-tumor activity for the study of cancer.		DUB
T3460	HhAntag		Hedgehog/Smoothened , Smo
	HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity.		Hedgehog/Smoothened , Smo
T15558	GSK319347A		IκB/IKK
	GSK319347A is a selective and potent dual inhibitor of TBK1 and IKKε with potential anti-tumor activity and inhibition of IKK2 activity, which can be used in the study of bladder cancer and lung adenocarcinoma.		IκB/IKK
T78650	Nrf2 activator-3		Antioxidant , Nrf2
	Nrf2 activator-3 is a potent Nrf2 activator with potential anti-inflammatory, antioxidant and anti-tumor activity, which can be used to study neurological and immune-related diseases.		Antioxidant , Nrf2
T13098	TBOPP		Others
	TBOPP is a selective DOCK1 inhibitor (IC50 : 8.4 μM), with anti-tumor activity for broader types of tumors.		Others
T60220	ROS kinases-IN-1		ROS Kinase
	ROS kinases-IN-1 is a ROS tyrosine kinase inhibitor with IC50 value of 1.22 μM. ROS kinases-IN-1 shows anti-tumor activity.		ROS Kinase
T10792L	CHK1-IN-4 hydrochloride	CHK1-IN-4 hydrochloride（2120398-41-4 Free base）	Chk
	CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1). CHK1-IN-4 hydrochloride potently inhibits chk1 phosphorylation in the tumor cells. CHK1-IN-4 hydrochloride has anti-tumor activity.		Chk
T22456	Voreloxin hydrochloride	SNS-595 hydrochloride,Vosaroxin	Apoptosis , Topoisomerase
	Voreloxin hydrochloride (SNS-595 hydrochloride) is a potent inhibitor of Topoisomerase II with broad-spectrum anti-tumor activity.		Apoptosis , Topoisomerase
T22231	Adenosine Dialdehyde (ADOX)	Periodate-oxidized adenosine,Adenosine, periodate oxidized,Adenox,Adenosinedialdehyde	Others
	Adenosine Dialdehyde (Periodate-oxidized adenosine) is a purine nucleoside analogue. Adenosine Dialdehyde is a potent inhibitor of S-Adenosylhomocysteine hydrolase (SAHH) (Ki=3.3 nM). Adenosine Dialdehyde exhibits potent...		Others
T77401	Bavituximab	Anti-PS MAb 3G4	Others
	Bavituximab (Anti-Human Phosphatidylserine Recombinant Antibody) is a monoclonal antibody against phosphatidylserine (PS) with vascular targeting and immunomodulatory properties. It can reactivate anti-tumor immunity to ...		Others
T60102L	Dimethylaminomicheliolide HCl		PKM
	Dimethylaminomicheliolide HCl has potential anti-inflammatory and anti-tumor activity and inhibits the proliferation of glioblastoma cells by targeting pyruvate kinase 2 (PKM2) and reconnecting aerobic cell populations.		PKM
T77582	Anti-inflammatory agent 51		NF-κB
	Anti-inflammatory agent 51 is an amide/sulfonamide derivative with anti-inflammatory and potentially anti-tumor activity and inhibition of NF-κB activation, which can be used to study acute lung injury and ulcerative col...		NF-κB
T10255	AES-135		HDAC
	AES-135 is a potent HDAC inhibitor, inhibits HDAC3, HDAC6, HDAC11 (IC50s: 654, 190, and 636 nM) with anti-tumor activity.		HDAC
T10468	Elimusertib hydrochloride(1876467-74-1 free base)	BAY-1895344 hydrochloride	ATM/ATR
	Elimusertib hydrochloride(1876467-74-1 free base) (BAY-1895344 hydrochloride) is a effective, orally available and selective ATR inhibitor with anti-tumor activity.		ATM/ATR
T50075	3,5-dimethyl-4-phenyl-1,2-oxazole		Others
	3,5-dimethyl-4-phenyl-1,2-oxazole is a heterocyclic compound used as a molecular structural unit. It has anti-inflammatory, anti-tumor, anti-bacterial and anti-fungal activity, as well as the ability to modulate the immu...		Others
T64295	Talotrexin ammonium		DHFR
	Talotrexin ammonium is a non-polyglutamic acid antifolate. Talotrexin ammonium inhibits tumor growth by targeting dihydrofolate reductase (DHFR), thereby improving anti-tumor activity in a wide range of cancer models, he...		DHFR
T77059	Leronlimab	PRO 140	CCR
	Leronlimab (PRO 140) is a humanized IgG4 anti-CCR5 monoclonal antibody. leronlimumab has both anti-HIV and anti-tumor activity, inhibiting CCR-mediated HIV-1 virus and cancer cell metastasis in mouse tumor models. Leronl...		CCR
T41345	AFMK	Formyl-N-acetyl-5-methoxykynurenamine,Acetyl-N-formyl-5-methoxykynurenamine	Apoptosis , Free radical scavengers , Antioxidant , Endogenous Metabolite
	AFMK (Formyl-N-acetyl-5-methoxykynurenamine) is an active metabolite of Melatonin with antioxidant and free radical scavenging activity. AFMK is a modulator of apoptosis and improves the anti-tumor effect of Gemcitabine ...
T7122	AZD-7648		DNA-PK
	AZD-7648 is an inhibitor of DNA-dependent protein kinase (DNA-PK) with the IC50 of 0.63 nM in an enzyme assay,has anti-tumor activity.		DNA-PK
T9127	MYLS22		Others
	MYLS22 is a first-in-class and selective inhibitor of optic atrophy 1 (OPA1) . MYLS22 can target endothelial OPA1 to curtail tumor growth and inhibits angiogenesis by impinging on NFkB activity and on angiogenic gene exp...		Others
T6891	MK-4101		Apoptosis , Hedgehog/Smoothened , Smo
	MK-4101, an effective inhibitor of the Hedgehog pathway, has anti-tumor activity through the induction of extensive apoptosis and inhibition of proliferation in tumor cells.		Apoptosis , Hedgehog/Smoothened , Smo
T10728	AS-0141	Cdc7-IN-6,PNT-141,SRA-141	CDK
	AS-0141 (Cdc7-IN-6) is a potent Cdc7 kinase inhibitor (IC50=4 nM) with anti-tumor activity.		CDK

Compounds

Target: Microtubule Associated

Uzansertib phosphate

T12477

Synonym: INCB053914 phosphate

Target: VEGFR, FLT, c-RET, PDGFR, Aurora Kinase

Buclizine dihydrochloride

T6426

Synonym: Longifene,Buclina,Buclizine HCl,UCB-4445

Target: 5-HT Receptor, AChR, Histamine Receptor

Zosuquidar trihydrochloride

T6018

Synonym: Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride

N-Acetyl-Calicheamicin

T12140

Synonym: N-Acetyl-Calicheamicin γ,N-Acetyl-γ-calicheamicin

Target: Antibacterial

Synonym: CS-045,Romozin,Rezulin,Romglizone,Noscal,Prelay

Target: Apoptosis, Ferroptosis, PPAR, Autophagy

Dehydroabiethylamine

T19783

Synonym: NSC-2955,NSC 2955,Dehydroabietylamine,NSC2955,Leelamine free base,Leelamine

Target: Others, Antibacterial, Antibiotic

2'-Deoxy-2'-fluoroarabinoadenosine

TNU0085

Synonym:

Target: Nucleoside Antimetabolite/Analog

Target: Dehydrogenase

Phenformin

T20158

Synonym: Debeone,N-Phenethylbiguanide,Insoral,BRN 1977317,Azucaps

KRAS G12C inhibitor 19

Synonym: KRAS G12D inhibitor 18,KRAS G12D IN 18

Target: Others, Ferroptosis, Nrf2

Synonym: 4-((3-Chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl acetate

Target: Serine/threonin kinase

Target: Gamma-secretase

Target: Hedgehog/Smoothened, Smo

Target: Antioxidant, Nrf2

CHK1-IN-4 hydrochloride

T10792L

Synonym: CHK1-IN-4 hydrochloride（2120398-41-4 Free base）

Target: Chk

Voreloxin hydrochloride

T22456

Synonym: SNS-595 hydrochloride,Vosaroxin

Target: Apoptosis, Topoisomerase

Adenosine Dialdehyde (ADOX)

T22231

Synonym: Periodate-oxidized adenosine,Adenosine, periodate oxidized,Adenox,Adenosinedialdehyde

Target: Others

Bavituximab

T77401

Synonym: Anti-PS MAb 3G4

Target: Others

Dimethylaminomicheliolide HCl

T60102L

Synonym:

Target: PKM

Anti-inflammatory agent 51

Elimusertib hydrochloride(1876467-74-1 free base)

T10468

Synonym: BAY-1895344 hydrochloride

Target: ATM/ATR

3,5-dimethyl-4-phenyl-1,2-oxazole

Synonym: Formyl-N-acetyl-5-methoxykynurenamine,Acetyl-N-formyl-5-methoxykynurenamine

Target: Apoptosis, Free radical scavengers, Antioxidant, Endogenous Metabolite

Target: Apoptosis, Hedgehog/Smoothened, Smo

AS-0141

T10728

Synonym: Cdc7-IN-6,PNT-141,SRA-141

Target: CDK

カタログ番号	製品名	別名	ターゲット
T9135	Epirosmanol		Others
	Epirosmanol is a diterpenoid containing a lactone moiety. Epirosmanol is a very weakly basic (essentially neutral) compound (based on its pKa).		Others
T5S0106	Peimisine	Ebeiensine	RAAS , AChR
	1. Peimisine (Ebeiensine) can affect M-receptor, excit β-receptor, restrain the release of internal calcium, and promote to releaseing nitrogen monoxidum in order to relax tracheal smooth muscle and relieve asthma. 2. Pe...		RAAS , AChR
TN2356	Tetradehydropodophyllotoxin	Dehydropodophyllotoxin	Others , Antifungal
	Tetradehydropodophyllotoxin (Dehydropodophyllotoxin) has anti-tumor activity.		Others , Antifungal
T4745	4-Carboxyquinoline	QUINOLINE-4-CARBOXYLIC ACID,4-Quinolinecarboxylic acid	Others , Endogenous Metabolite
	4-Carboxyquinoline (4-Quinolinecarboxylic acid) showed anti-tumor activity against L1210 leukemia and B16 melanoma.		Others , Endogenous Metabolite
TN1531	Cratoxylone		Antifungal
	Cratoxylone is derived from the bark of the Cochin tree and has anti-plasmodial activity and potential anti-tumor and antioxidant activity.		Antifungal
T5726	Specneuzhenide	Nuezhenide	Others
	Specneuzhenide (Nuezhenide) is a phenol glycoside isolated from Ligustrum sinense. Specneuzhenide (Nuezhenide) possesses anti-tumor activity,has anti-angiogenic and vision improvement effects.		Others
T8271	10Z-Nonadecenoic acid		Endogenous Metabolite
	10Z-Nonadecenoic acid is a long-chain fatty acid with anti-tumor activity.		Endogenous Metabolite
TN4991	Senkyunolide A		Others
	Senkyunolide A is a natural product isolated from Ligusticum chuanxiong Hort, with anti-tumor activity.		Others
T8169	Decursinol		Others
	Decursinol is isolated from the roots of Angelica Gigas with an antinociceptive effect. It also has anti-tumor and anti-metastasis activity.		Others
TN2337	Poricoic acid AM
	Poricoic acid AM is a triterpenoid compound extracted from Poria cocos, demonstrating anti-tumor activity.
T10117	3'-O-Acetylhamaudol		Others
	3'- O- Acetylhamaudol, isolated from the roots of Angelica japonica, exhibits anti-tumor activity through dual actions, anti-angiogenesis and intestinal intraepithelial lymphocyte activation.		Others
T3400	Bakuchiol		p38 MAPK , DNA/RNA Synthesis , Autophagy
	Bakuchiol possesses anti-tumor,and anti-helmenthic properties. It has cytotoxic activity, mainly due to its DNA polymerase1 inhibiting activity. Bakuchiol has anti-bacterial activity against oral pathogens, has great pot...		p38 MAPK , DNA/RNA Synthesis , Autophagy
T4S1519	Pseudoginsenoside RT5		Others
	1. Pseudoginsenoside RT5 has anti-epilepsy, anti-depressant activity by promoting nerve growth and improve cognitive ability. 2. Pseudoginsenoside RT5 has anti-bacterial, anti-tumor and anti-malaria activities.		Others
TN1557	Decursinol angelate		ERK , VEGFR , PKC , JNK
	Decursinol angelate has anti-tumor, anti-inflammatory, anti-oxidant, and hepatoprotective activities, it inhibits VEGF-induced angiogenesis via suppression of the VEGFR-2-signaling pathway; it also suppresses invasion an...		ERK , VEGFR , PKC , JNK
TN1459	Bufarenogin	3beta,12beta,14-Trihydroxy-11-oxo-5beta-bufa-20,22-dienolide	ERK , MEK , PI3K
	Bufarenogin (3beta,12beta,14-Trihydroxy-11-oxo-5beta-bufa-20,22-dienolide) is a bufadienolide isolated from parotoid gland secretions of the Cuban endemic toad Peltophryne fustiger. Bufarenogin shows anti-tumor activity.		ERK , MEK , PI3K
TQ0118	Britannilactone	Desacetylinulicin	Others
	Britannilactone (Desacetylinulicin) is a sesquiterpene from Inula britannica with anti-inflammatory and anti-tumor activity.Britannilactone has been associated with this antimelanotic activity and can be used in studies ...		Others
T3S1513	(20R)-Protopanaxadiol	Protopanaxadiol,20R-Protopanaxadiol,(20R)-Protopanaxdiol	Others , Antibacterial
	1. (20R)-Protopanaxadiol ((20R)-Protopanaxdiol) has the effect of anti-tumor through increasing the activity of body immunity, inhibiting tumor interstitial microvascular density and its proliferation activity, improving...		Others , Antibacterial
T3S0872	Paederoside		Antiviral , HBV
	1. Paederoside is a potent deterrent against the beetle was isolated from the aphid . 2. Paederoside displays high anti-tumor promoting activity against the Epstein-Barr virus activation.		Antiviral , HBV
T5S1882	Songorine	Napellonine,Zongorine,Bullatine G	Others , GABA Receptor
	Songorine (Napellonine) shows favorable anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.		Others , GABA Receptor
T7984	2-Hydroxyflavanone		Others
	2-Hydroxyflavanone is a naturally occurring flavonoid found in many plants and fruits. It has antioxidant, anti-inflammatory and anti-tumor activity, scavenging free radicals, reducing inflammation and inhibiting the gro...		Others
T3S0895	Spirostan-3-ol	Sarsaponin	Others
	Spirostan-3-ol (Sarsaponin) is a stereoisomer of Sarsasapogenin (S142505), a steroid glycoside isolated from plant materials. A saponin with with potential anti-tumor activity via apoptosis.		Others
T5660	Menthone		IL Receptor , TNF , NF-κB , Parasite
	Menthone has anti-inflammary activity,, it can suppress the lipopolysaccharide (LPS)-induced proinflammatory cytokines, interleukin-1beta (IL-1beta) and tumor necrosis factor-alpha (TNF-alpha),as well as nuclear factor k...		IL Receptor , TNF , NF-κB , Parasite
T4S21320	ISOGINKGETIN	4',4'''-Dimethylamentoflavone	MMP , Others
	1. ISOGINKGETIN (4',4'''-Dimethylamentoflavone), a compound derived from the leaves of Ginkgo biloba, to up-regulate adiponectin secretion with potency comparable to that of rosiglitazone, a known modulator of adiponecti...		MMP , Others
T0968	Paclitaxel	Taxol,NSC 125973	Apoptosis , Microtubule Associated , Autophagy
	Paclitaxel (Taxol) is a natural product and a microtubule polymer stabilizer. Paclitaxel has anti-tumor activity and causes cell death by inducing mitotic arrest, apoptosis, and cell autophagy.		Apoptosis , Microtubule Associated , Autophagy
T15705	Laminaran	β-1,3-Glucan
	Laminaran is a β-1,3-glucan isolated from brown algae, often serving as a typical ligand for Dectin-1. It possesses anti-cancer, immune-modulating, and radiation-protective properties. Laminaran can be catalyzed by gluca...
TN1516	Cnidicin		NOS , NO Synthase
	Cnidicin has anti-allergic and anti-inflammatory activity, it inhibits the degranulation of mast cell and the NO generation in RAW 264.7 cells(IC50 value, 7.5 microM). Cnidicin exhibits a significant inhibition on the pr...		NOS , NO Synthase
T7990	9-hydroxy-4-androstene-3,17-dione		Others
	9-hydroxy-4-androstene-3,17-dione is a steroid hormone. It has anti-tumor activity and can inhibit the growth of many types of cancer cells, including breast, prostate and lung cancer cells.		Others
T13818	Phytohemagglutinin	PHA-M	Apoptosis
	Phytohemagglutinin (PHA-M) is a lectin, isolated from the red kidney bean , induces apoptosis via increasing proapoptotic protein Bax and activating caspases-3. Anti-tumor activity		Apoptosis
TN7052	Crocin III	Crocetin-mono-(β-D-gentiobiosyl)-ester	Others
	Crocin III (Crocetin-mono-(β-D-gentiobiosyl)-ester) is a crocin derived from saffron (Crocus sutivus L.). Crocins inhibit the cell growth of tumor cells and have anti-inflammatory activity.		Others
T6S0117	Avicularin	Fenicularin	ERK
	Avicularin (Fenicularin) has anti-allergic, anti-inflammatory, hepatoprotective, antioxidant, anti-tumor and other activities. It ameliorates human hepatocellular carcinoma by modulating the activities of NF-κB(p65), COX...		ERK
T3S1641	Esculentoside H		TNF , NF-κB , JNK
	Phytolaccaceae has anti-tumor activity, the mechanism may be related to the capacity of Esculentoside H for TNF release.		TNF , NF-κB , JNK
TN1661	Ganoderic acid C2		Reductase , Histamine Receptor , Immunology/Inflammation related
	Ganoderic acid C2 has anti-inflammatory,and anti-tumor-promoting activities. Ganoderic acid C2 can inhibit histamine release, it also has inhibitory effects on the induction of Epstein-Barr Virus early antigen.
Fr12277	4-Hydroxy-6-methylcoumarin		Others
	4-Hydroxy-6-methylcoumarin (4-HMC) is a naturally occurring phenolic compound, a derivative of coumarin, found in a variety of plants, fungi, and bacteria. It has anti-inflammatory and anti-tumor activity.4-HMC is used a...		Others
T1034	Docetaxel	NSC 628503,RP-56976	Apoptosis , Microtubule Associated , Endogenous Metabolite
	Docetaxel (RP-56976) is a semi-synthetic analog of paclitaxel, a microtubule depolymerization inhibitor (IC50=0.2 μM). Docetaxel attenuates the effects of bcl-2 and bcl-xL gene expression and exhibits apoptosis-inducing,...		Apoptosis , Microtubule Associated , Endogenous Metabolite
T36715	Tetrac	Tetraiodothyroacetic acid,3,3',5,5'-Tetraiodothyroacetic acid	Apoptosis , EGFR
	Tetrac (Tetraiodothyroacetic acid) is a derivative of L-thyroxine (T4), a thyroxine integrin receptor antagonist.Tetrac induces antiproliferation by blocking EGFR-mediated cell signaling in colorectal cancer cells.Tetrac...		Apoptosis , EGFR
T6S1579	Monotropein	Monotropeine	Others
	1. Monotropein (Monotropeine) has antinociceptive action. 2. Monotropein has anti-apoptosis and anti-catabolic activity in chondrocytes. 3. Monotropein has anti-inflammatory action by inhibition of the expressions of inf...		Others
T3897	Isoschaftoside		Anti-infection , Antifungal
	Isoschaftoside is used as an intercrop due to its allelopathic inhibition of parasitism by Striga hermonthica, an obligate parasitic weed that can devastate the maize crop. Isoschaftoside has anti-tumor, antioxidant, and...		Anti-infection , Antifungal
T3S0737	Flavokawain A	Flavokavain A	Apoptosis , p38 MAPK
	NSC-37445 has anti-tumor activity, such as inhibits growth of bladder tumor cells in a nude mice model , prevents the recurrence and progression of non-muscle-invasive urothelial cell carcinoma. NSC-37445 can significant...		Apoptosis , p38 MAPK
T2P2806	Hederacolchiside A1	Raddeanoside R13	Apoptosis , ERK , MEK , Akt , PI3K , Parasite , mTOR
	Hederacolchiside A1 (Raddeanoside R13) shows anti-leishmanial activity, it exhibits a strong antiproliferative activity on all stages of development of the parasite by altering membrane integrity and potential. Hederacol...		Apoptosis , ERK , MEK , Akt , PI3K , Parasite , mTOR
T2978	Mogroside V		AMPK
	Mogroside V is a widely used sweetener, has in vitro AMPK activating effect, it also has anti-inflammatory potential in murine macrophages and a murine ear edema model, and has the potential to protect against LPS-induce...		AMPK
T6S0119	Dauricine		Apoptosis , Others , NF-κB
	1. Dauricine has pulmonary toxicity, can produce pulmonary injury in CD-1 mice by the metabolism of Dauricine mediated by CYP3A. 2. Dauricinec can pass the blood-brain barrier, and that P-glycoprotein has an important ro...		Apoptosis , Others , NF-κB
T4672	Brevilin A		Apoptosis , Anti-infection , JAK , STAT , Autophagy
	Brevilin A is a sesquiterpene lactone isolated from Centipeda minima, inhibits janus kinase activity and blocks STAT3 signaling in cancer cells with anti-tumor activity. Brevilin A is a selective inhibitor of JAK-STAT si...		Apoptosis , Anti-infection , JAK , STAT , Autophagy
T6S1256	Ruscogenin		NOS , NF-κB , NOD-like Receptor (NLR)
	1. Ruscogenin has anti-inflammatory activity, suppressed zymosan A-evoked peritoneal total leukocyte migration in mice in a dose-dependent manner, 2. Ruscogenin inhibited adhesion of leukocytes to a human umbilical vein ...		NOS , NF-κB , NOD-like Receptor (NLR)
TN1564	Delphinidin 3-glucoside chloride	Delphinidin-3-O-glucoside chloride	Apoptosis , EGFR
	Delphinidin 3-glucoside chloride (Delphinidin-3-O-glucoside chloride) is a dietary phenolic substance found in Hibiscus sabdariffa extracts. Delphinidin 3-glucoside chloride has antioxidant activity, induces pro-apoptoti...		Apoptosis , EGFR
TMA2008	3-Hydroxy-1,5-diphenyl-1-pentanone
	(+)-3-Hydroxy-1,5-diphenyl-1-pentanone exhibits both immunomodulatory and anti-tumor activity.
T14330	Ascochlorin	Ilicicolin D	STAT
	Ascochlorin (Ilicicolin D), an isoprenoid antibiotic, primarily exerts its anti-tumor properties by inhibiting the STAT3 signaling pathway. It induces apoptosis and possesses anti-inflammatory activity[1][2][3].		STAT
TN2926	3-Epicabraleahydroxylactone		Others
	3-Epicabraleahydroxylactone has anti-tumor promoting effect, it has anti-carcinogenic activity by the inhibitory effect on the induction of Epstein-Barr virus early antigen(EBV-EA) by the tumor promoter.		Others
T12093	Monascin		Others
	Monascin is a kind of azaphilonoid pigments extracted from Monascus pilosus-fermented rice (red-mold rice),exhibits anti-tumor-initiating activity and anti-inflammatory activity .		Others
T20320	Tristearin	Glyceryl tristearate,Stearin,Glycowax S 932,Trioctadecanoin,Glycerol tristearate	Others
	Tristearin (Glycerol tristearate) is a natural product isolated from the leaves and stems of Hoag's Hooker with anti-tumor activity.		Others
TMA2576	Episappanol		IL Receptor , TNF
	Episappanol has anti-inflammatory activity , it can significantly inhibit the secretion of the pro-inflammatory cytokines interleukin (IL-6) and tumor necrosis factor-alpha (TNF-α).		IL Receptor , TNF
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天然物製品

Tetradehydropodophyllotoxin

TN2356

Synonym: Dehydropodophyllotoxin

Target: Others, Antifungal

4-Carboxyquinoline

T4745

Synonym: QUINOLINE-4-CARBOXYLIC ACID,4-Quinolinecarboxylic acid

Target: Others, Endogenous Metabolite

10Z-Nonadecenoic acid

T8271

Synonym:

Target: Endogenous Metabolite

Target: p38 MAPK, DNA/RNA Synthesis, Autophagy

Pseudoginsenoside RT5

Target: ERK, VEGFR, PKC, JNK

Bufarenogin

TN1459

Synonym: 3beta,12beta,14-Trihydroxy-11-oxo-5beta-bufa-20,22-dienolide

Target: ERK, MEK, PI3K

Britannilactone

TQ0118

Synonym: Desacetylinulicin

Target: Others

(20R)-Protopanaxadiol

T3S1513

Synonym: Protopanaxadiol,20R-Protopanaxadiol,(20R)-Protopanaxdiol

Target: Others, Antibacterial

Paederoside

T3S0872

Synonym:

Target: Antiviral, HBV

Songorine

T5S1882

Synonym: Napellonine,Zongorine,Bullatine G

Target: Others, GABA Receptor

Target: IL Receptor, TNF, NF-κB, Parasite

ISOGINKGETIN

T4S21320

Synonym: 4',4'''-Dimethylamentoflavone

Target: MMP, Others

Paclitaxel

T0968

Synonym: Taxol,NSC 125973

Target: Apoptosis, Microtubule Associated, Autophagy

Laminaran

T15705

Synonym: β-1,3-Glucan

Target: NOS, NO Synthase

9-hydroxy-4-androstene-3,17-dione

Synonym: Crocetin-mono-(β-D-gentiobiosyl)-ester

Target: TNF, NF-κB, JNK

Ganoderic acid C2

TN1661

Synonym:

Target: Reductase, Histamine Receptor, Immunology/Inflammation related

4-Hydroxy-6-methylcoumarin

Synonym: NSC 628503,RP-56976

Target: Apoptosis, Microtubule Associated, Endogenous Metabolite

Tetrac

T36715

Synonym: Tetraiodothyroacetic acid,3,3',5,5'-Tetraiodothyroacetic acid

Target: Apoptosis, EGFR

Monotropein

T6S1579

Synonym: Monotropeine

Target: Anti-infection, Antifungal

Flavokawain A

T3S0737

Synonym: Flavokavain A

Target: Apoptosis, p38 MAPK

Hederacolchiside A1

T2P2806

Synonym: Raddeanoside R13

Target: Apoptosis, ERK, MEK, Akt, PI3K, Parasite, mTOR

Target: Apoptosis, Others, NF-κB

Brevilin A

T4672

Synonym:

Target: Apoptosis, Anti-infection, JAK, STAT, Autophagy

Ruscogenin

T6S1256

Synonym:

Target: NOS, NF-κB, NOD-like Receptor (NLR)

Delphinidin 3-glucoside chloride

TN1564

Synonym: Delphinidin-3-O-glucoside chloride

Target: Apoptosis, EGFR

3-Hydroxy-1,5-diphenyl-1-pentanone

Synonym: Ilicicolin D

Target: STAT

3-Epicabraleahydroxylactone

Synonym: Glyceryl tristearate,Stearin,Glycowax S 932,Trioctadecanoin,Glycerol tristearate

Target: IL Receptor, TNF

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Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-04552	AKT1 Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	v-akt murine thymoma viral oncogene homolog 1 (AKT1), or protein kinase B-alpha (PKB-ALPHA) is a serine-threonine protein kinase, belonging to the Protein Kinase Superfamily. AKT1 is a major mediator of the responses to ...
TMPY-06983	IFN gamma Protein, Human, Recombinant (E. coli)	Human	E. coli
	IFN gamma, also known as IFNG, is a secreted protein that belongs to the type II interferon family. IFN gamma is produced predominantly by natural killer and natural killer T cells as part of the innate immune response, ...
TMPH-02591	COL4A3 Protein, Mouse, Recombinant (His & Myc)	Mouse	E. coli
	Type IV collagen is the major structural component of glomerular basement membranes (GBM), forming a 'chicken-wire' meshwork together with laminins, proteoglycans and entactin/nidogen.; Tumstatin, a cleavage fragment cor...
TMPK-00948	CDH17 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-00952	CDH17 Domain 3 & 4 Protein, Human, Recombinant (mFc)	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-01224	CDH17 Protein (Primary Amine Labeling), Mouse, Recombinant (His), Biotinylated	Mouse	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-00555	CDH17 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-00473	CDH17 Protein, Rhesus macaque, Recombinant (His)	Rhesus	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPH-02590	COL4A2 Protein, Mouse, Recombinant (His)	Mouse	E. coli
	Type IV collagen is the major structural component of glomerular basement membranes (GBM), forming a 'chicken-wire' meshwork together with laminins, proteoglycans and entactin/nidogen.; Canstatin, a cleavage product corr...
TMPK-00947	CDH17 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-00950	CDH17 Domain 6-7 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-01223	CDH17 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-00953	CDH17 Domain 6-7 Protein, Human, Recombinant (mFc)	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-00949	CDH17 Domain 7 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-00951	CDH17 Domain 5-7 Protein (Primary Amine Labeling), Human, Recombinant (His), Biotinylated	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPH-01112	COL4A1 Protein, Human, Recombinant (GST)	Human	E. coli
	Type IV collagen is the major structural component of glomerular basement membranes (GBM), forming a 'chicken-wire' meshwork together with laminins, proteoglycans and entactin/nidogen.; Arresten, comprising the C-termina...
TMPJ-00766	ANXA1 Protein, Human, Recombinant	Human	E. coli
	Annexin A1 is the first characterized member of the annexin family of proteins and is able to bind to cellular membranes in a calcium-dependent manner, promoting membrane fusion and endocytosis. Annexin A1 has anti-infla...
TMPJ-00948	Endostatin Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Endostatin, an endogenous non‑glycosylated inhibitor of endothelial cell proliferation and angiogenesis. It is produced and/or trimmed by metalloproteinases such as MMP‑2 and MMP‑9, and cathepsins S, B and L. The N‑termi...
TMPY-00186	GHRH Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	The role of hypothalamic growth hormone-releasing hormone (GHRH) in the release of growth hormone (GH) from the pituitary is well established. Extra-hypothalamic growth hormone-releasing hormone (GHRH) plays an important...
TMPH-01552	IRF1 Protein, Human, Recombinant (GST & His)	Human	Baculovirus Insect Cells
	Transcriptional regulator which displays a remarkable functional diversity in the regulation of cellular responses. Regulates transcription of IFN and IFN-inducible genes, host response to viral and bacterial infections,...
TMPJ-00189	TIM-3/KIM-3/HAVCR2 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	T cell immunoglobulin and mucin domain 3 is a member of the TIM family of immune regulating molecules. Mature cynomolgus TIM3 consists of a 182 amino acid (aa)extracellular domain (ECD), a 21 aa transmembrane segment, an...
TMPY-01909	Elafin Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Elafin, also known as Elastase-specific inhibitor, Peptidase inhibitor 3, Protease inhibitor WAP3, Skin-derived antileukoproteinase, WAP four-disulfide core domain protein 14, PI3, WAP3 and WFDC14, is a secreted protein ...
TMPY-02084	Thioredoxin 2/TRX2 Protein, Human, Recombinant (His)	Human	E. coli
	Thioredoxin-2, also known as TXN2, MTRX and TRX2, is a member of the thioredoxin family. Tryparedoxins (TXN) are thioredoxin-related proteins which, as trypanothione:peroxiredoxin oxidoreductases, constitute the trypanot...
TMPH-03753	MYLK Protein, Human, Recombinant (His)	Human	E. coli
	Calcium/calmodulin-dependent myosin light chain kinase implicated in smooth muscle contraction via phosphorylation of myosin light chains (MLC). Also regulates actin-myosin interaction through a non-kinase activity. Phos...

AKT1 Protein, Human, Recombinant (His)

TMPY-04552

Species: Human

Expression System: Baculovirus Insect Cells

IFN gamma Protein, Human, Recombinant (E. coli)

TMPY-06983

Species: Human

Expression System: E. coli

COL4A3 Protein, Mouse, Recombinant (His & Myc)

TMPH-02591

Species: Mouse

Expression System: E. coli

CDH17 Protein, Human, Recombinant (hFc)

TMPK-00948

Species: Human

Expression System: HEK293 Cells

CDH17 Domain 3 & 4 Protein, Human, Recombinant (mFc)

TMPK-00952

Species: Human

Expression System: HEK293 Cells

CDH17 Protein (Primary Amine Labeling), Mouse, Recombinant (His), Biotinylated

TMPK-01224

Species: Mouse

Expression System: HEK293 Cells

CDH17 Protein, Cynomolgus, Recombinant (His)

TMPK-00555

Species: Cynomolgus

Expression System: HEK293 Cells

CDH17 Protein, Rhesus macaque, Recombinant (His)

TMPK-00473

Species: Rhesus

Expression System: HEK293 Cells

COL4A2 Protein, Mouse, Recombinant (His)

TMPH-02590

Species: Mouse

Expression System: E. coli

CDH17 Protein, Human, Recombinant (His & Avi), Biotinylated

TMPK-00947

Species: Human

Expression System: HEK293 Cells

CDH17 Domain 6-7 Protein, Human, Recombinant (hFc)

TMPK-00950

Species: Human

Expression System: HEK293 Cells

CDH17 Protein, Mouse, Recombinant (His)

TMPK-01223

Species: Mouse

Expression System: HEK293 Cells

CDH17 Domain 6-7 Protein, Human, Recombinant (mFc)

TMPK-00953

Species: Human

Expression System: HEK293 Cells

CDH17 Domain 7 Protein, Human, Recombinant (hFc)

TMPK-00949

Species: Human

Expression System: HEK293 Cells

CDH17 Domain 5-7 Protein (Primary Amine Labeling), Human, Recombinant (His), Biotinylated

TMPK-00951

Species: Human

Expression System: HEK293 Cells

COL4A1 Protein, Human, Recombinant (GST)

TMPH-01112

Species: Human

Expression System: E. coli

ANXA1 Protein, Human, Recombinant

TMPJ-00766

Species: Human

Expression System: E. coli

Endostatin Protein, Mouse, Recombinant (His)

TMPJ-00948

Species: Mouse

Expression System: HEK293 Cells

GHRH Protein, Human, Recombinant (hFc)

TMPY-00186

Species: Human

Expression System: HEK293 Cells

IRF1 Protein, Human, Recombinant (GST & His)

TMPH-01552

Species: Human

Expression System: Baculovirus Insect Cells

TIM-3/KIM-3/HAVCR2 Protein, Cynomolgus, Recombinant (His)

TMPJ-00189

Species: Cynomolgus

Expression System: HEK293 Cells

Elafin Protein, Human, Recombinant (His)

TMPY-01909

Species: Human

Expression System: HEK293 Cells

Thioredoxin 2/TRX2 Protein, Human, Recombinant (His)

TMPY-02084

Species: Human

Expression System: E. coli

MYLK Protein, Human, Recombinant (His)

TMPH-03753

Species: Human

Expression System: E. coli

カタログ番号	製品名
L2100	Anti-Cancer Compound Library	7234 compounds
	A unique collection of 7234 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L2160	Anti-Cancer Active Compound Library	3188 compounds
	A unique collection of 3188 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L2130	Anti-Cancer Metabolism Compound Library	1268 compounds
	A unique collection of 1268 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS);
L6120	Flavonoid Natural Product Library	514 compounds
	A unique collection of 514 flavonoids can be used for high throughput and high content screening；
L2196	Anti-Ovarian Cancer Compound Library	1867 compounds

ライブラリー

Anti-Cancer Compound Library

L2100

Compounds: 7234

Anti-Cancer Active Compound Library

L2160

Compounds: 3188

Anti-Cancer Metabolism Compound Library

L2130

Compounds: 1268

Flavonoid Natural Product Library

L6120

Compounds: 514

Anti-Ovarian Cancer Compound Library

L2196

Compounds: 1867